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NF-56-EJ40 hydrochloride
CAS No. 2728500-80-7
NF-56-EJ40 hydrochloride ( —— )
产品货号. M33038 CAS No. 2728500-80-7
NF-56-EJ40 hydrochloride is a potent, high-affinity, and highly selective human SUCNR1 (GPR91) antagonist with an IC50 of 25 nM and a Ki of 33 nM, and shows almost no activity towards rat SUCNR1. NF-56-EJ40 hydrochloride has high affinity for humanized rat SUCNR1 with a Ki value of 17.4 nM.
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 5MG | ￥404 | 有现货 |
|
| 10MG | ￥606 | 有现货 |
|
| 25MG | ￥1001 | 有现货 |
|
| 50MG | ￥1501 | 有现货 |
|
| 100MG | ￥2196 | 有现货 |
|
| 200MG | ￥3297 | 有现货 |
|
| 500MG | 获取报价 | 有现货 |
|
| 1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称NF-56-EJ40 hydrochloride
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注意事项本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
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产品简述NF-56-EJ40 hydrochloride is a potent, high-affinity, and highly selective human SUCNR1 (GPR91) antagonist with an IC50 of 25 nM and a Ki of 33 nM, and shows almost no activity towards rat SUCNR1. NF-56-EJ40 hydrochloride has high affinity for humanized rat SUCNR1 with a Ki value of 17.4 nM.
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产品描述NF-56-EJ40 hydrochloride is a potent, high-affinity, and highly selective human SUCNR1 (GPR91) antagonist with an IC50 of 25 nM and a Ki of 33 nM, and shows almost no activity towards rat SUCNR1. NF-56-EJ40 hydrochloride has high affinity for humanized rat SUCNR1 with a Ki value of 17.4 nM.
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体外实验——
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体内实验——
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同义词——
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通路GPCR/G Protein
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靶点GHSR
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受体GHSR
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研究领域——
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适应症——
化学信息
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CAS Number2728500-80-7
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分子量516.46
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分子式C27H31Cl2N3O3
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纯度>98% (HPLC)
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溶解度——
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SMILESO=C(CC1=C(NC(C2=CC=CC(C3=CC=C(CN4CCN(CC4)C)C=C3)=C2)=O)C=CC=C1)O.Cl.Cl
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化学全称——
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
产品手册
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